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Most polar substances are readily dissolved in aqueous media (i. e. , are hydrophilic) and lipophilic ones in apolar media.
According to the chemical structure of the side chain, phenothiazines and thioxanthenes can be subdivided into aliphatic (chlorpromazine, triflupromazine, p. 239 and piperazine congeners (trifluperazine, fluphenazine, flupentixol, p. 239). The antipsychotic effect is probably due to an antagonistic action at dopamine receptors. |
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