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When intake stops, nicotine concentration in plasma shows an initial rapid fall, reflecting distribution into tissues, and a terminal elimination phase with a half-life of 2 h. Nicotine is degraded by oxidation.
Its congener, dihydroergotamine, is furthermore employed in orthostatic complaints. Other lysergic acid derivatives are the 5-HT antagonist methysergide, the dopamine agonists bromocriptine, pergolide, and cabergolide, and the hallucinogen lysergic acid diethylamide (LSD). |
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